h1 receptor agonist

C3a Receptor Agonist

MBS5798977-5mg 5(mg
EUR 605

C3a Receptor Agonist

T38287-10mg 10mg Ask for price
Description: C3a Receptor Agonist

C3a Receptor Agonist

T38287-1g 1g Ask for price
Description: C3a Receptor Agonist

C3a Receptor Agonist

T38287-1mg 1mg Ask for price
Description: C3a Receptor Agonist

C3a Receptor Agonist

T38287-50mg 50mg Ask for price
Description: C3a Receptor Agonist

C3a Receptor Agonist

T38287-5mg 5mg Ask for price
Description: C3a Receptor Agonist

TGR5 Receptor Agonist

1722-5 each
EUR 405.6

TGR5 Receptor Agonist

B1185-10 10 mg
EUR 222.4
Description: Others|Others

TGR5 Receptor Agonist

B1185-100 100mg
EUR 1320
Description: Others|Others

TGR5 Receptor Agonist

B1185-25 25 mg
EUR 686.4
Description: TGR5 Receptor Agonist is a potent and selective agonist of TGR5 G-protein receptor with a pEC50 value of 6.8 in the U2-OS cell assay [1].

TGR5 Receptor Agonist

B1185-5 5 mg
EUR 132
Description: Others|Others

TGR5 Receptor Agonist

B1185-50 50mg
EUR 413.6
Description: Others|Others

TGR5 Receptor Agonist

MBS130022-100mg 100mg
EUR 1065

TGR5 Receptor Agonist

MBS130022-500mg 500mg
EUR 2775

TGR5 Receptor Agonist

HY-14229 100mg
EUR 630.96
Description: TGR5 Receptor Agonist (CCDC), a potent Takeda G protein-coupled receptor 5 (TGR5; GPCR19) agonist, shows improved potency in the U2-OS cells and melanophore cells with pEC50s of 6.8 and 7.5, respectively. TGR5 Receptor Agonist can induce peripheral and central hypersensitivity to bladder distension in mice, and increase intracellular Ca2+ concentration. TGR5 Receptor Agonist can also reduces food intake and improves insulin responsiveness, in diet-induced obese mice. TGR5 Receptor Agonist can be used to research diabetes, bladder hypersensitivity and anti-obesity[1][2][3][4].

TGR5 Receptor Agonist

MBS576315-10mg 10mg
EUR 210

TGR5 Receptor Agonist

MBS576315-25mg 25mg
EUR 365

TGR5 Receptor Agonist

MBS576315-2mg 2mg
EUR 145

TGR5 Receptor Agonist

MBS576315-50mg 50mg
EUR 490

TGR5 Receptor Agonist

MBS576315-5mg 5mg
EUR 165

TGR5 Receptor Agonist

T1824-10mg 10mg Ask for price
Description: TGR5 Receptor Agonist

TGR5 Receptor Agonist

T1824-1g 1g Ask for price
Description: TGR5 Receptor Agonist

TGR5 Receptor Agonist

T1824-1mg 1mg Ask for price
Description: TGR5 Receptor Agonist

TGR5 Receptor Agonist

T1824-50mg 50mg Ask for price
Description: TGR5 Receptor Agonist

TGR5 Receptor Agonist

T1824-5mg 5mg Ask for price
Description: TGR5 Receptor Agonist

GPR120 receptor agonist

MBS3607893-100mg 100mg
EUR 1695

GPR120 receptor agonist

MBS3607893-10mg 10mg
EUR 515

GPR120 receptor agonist

MBS3607893-2mg 2mg
EUR 295

GPR120 receptor agonist

MBS3607893-50mg 50mg
EUR 1260

GPR120 receptor agonist

MBS3607893-5mg 5mg
EUR 400

GPR120 Receptor Agonist

MBS5750453-10mg 10mg
EUR 455

GPR120 Receptor Agonist

MBS5750453-1mg 1mg
EUR 175

GPR120 Receptor Agonist

MBS5750453-2mg 2mg
EUR 225

GPR120 Receptor Agonist

MBS5750453-50mg 50mg
EUR 1200

GPR120 Receptor Agonist

MBS5750453-5mg 5mg
EUR 335

THRβ receptor agonist-1

HY-153535 Get quote Ask for price
Description: THRβ receptor agonist-1 is a THRβ receptor agonist[1].

sst2 Receptor agonist-1

HY-110161 Get quote Ask for price
Description: sst2 Receptor agonist-1 is a potent somatostatin receptor subtype 2 (sst2) agonist with a Ki value of 0.025 nM and a cAMP IC50 value of 4.8 nM. sst2 Receptor agonist-1 can inhibit rat growth hormone (GH) secretion and ocular neovascular lesion formation. Antiangiogenic effect[1].

S1P5 receptor agonist-1

HY-148198 Get quote Ask for price
Description: S1P5 receptor agonist-1 (example 6) is a potent and selective agonist of S1P5 receptor with an EC50 value of 20 nM[1].

Thrombin Receptor Agonist

070-73 500 μg
EUR 114.48

Thrombin Receptor Agonist

MBS826474-10mg 10mg
EUR 480

Thrombin Receptor Agonist

MBS826474-1mg 1mg
EUR 185

Thrombin Receptor Agonist

MBS826474-5mg 5mg
EUR 325

Thrombin Receptor Agonist

MBS826474-5x10mg 5x10mg
EUR 2085

RXFP1 receptor agonist-1

HY-156536 Get quote Ask for price
Description: RXFP1 receptor agonist-1 (Example 2) is a RXFP1 receptor agonist. RXFP1 receptor agonist-1 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 300 nM[1].

RXFP1 receptor agonist-2

HY-156537 Get quote Ask for price
Description: RXFP1 receptor agonist-2 (Example 124) is a RXFP1 receptor agonist. RXFP1 receptor agonist-2 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1 nM[1].

RXFP1 receptor agonist-3

HY-156538 Get quote Ask for price
Description: RXFP1 receptor agonist-3 (Example 223) is a RXFP1 receptor agonist. RXFP1 receptor agonist-3 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 2 nM[1].

RXFP1 receptor agonist-4

HY-156539 Get quote Ask for price
Description: RXFP1 receptor agonist-4 (Example 268) is a RXFP1 receptor agonist. RXFP1 receptor agonist-4 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 4.9 nM[1].

RXFP1 receptor agonist-5

HY-156540 Get quote Ask for price
Description: RXFP1 receptor agonist-5 (Example 98) is a RXFP1 receptor agonist. RXFP1 receptor agonist-5 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1.3 nM[1].

RXFP1 receptor agonist-6

HY-156541 Get quote Ask for price
Description: RXFP1 receptor agonist-6 (Example 7) is a RXFP1 receptor agonist. RXFP1 receptor agonist-6 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 12 nM[1].

RXFP1 receptor agonist-7

HY-156542 Get quote Ask for price
Description: RXFP1 receptor agonist-7 (Example 2) is a RXFP1 receptor agonist. RXFP1 receptor agonist-7 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 4.2 nM[1].

RXFP1 receptor agonist-8

HY-156543 Get quote Ask for price
Description: RXFP1 receptor agonist-8 (Example 2) is a RXFP1 receptor agonist. RXFP1 receptor agonist-8 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1.8 nM[1].

GP130 receptor agonist-1

HY-121488 1 mg
EUR 519.49
Description: GP130 receptor agonist-1 is a potent, brain-penetrant and orally active GP130 receptor agonist. GP130 receptor agonist-1 has a neuroprotective effect on NMDA-induced neurotoxicity[1].

GP130 receptor agonist-1

T9157-10mg 10mg Ask for price
Description: GP130 receptor agonist-1

GP130 receptor agonist-1

T9157-1g 1g Ask for price
Description: GP130 receptor agonist-1

GP130 receptor agonist-1

T9157-1mg 1mg Ask for price
Description: GP130 receptor agonist-1

GP130 receptor agonist-1

T9157-50mg 50mg Ask for price
Description: GP130 receptor agonist-1

GP130 receptor agonist-1

T9157-5mg 5mg Ask for price
Description: GP130 receptor agonist-1

GPR109 receptor agonist-1

HY-107580 10 mg
EUR 194.81
Description: GPR109 receptor agonist-1 (Compound 3a) is a highly selective agonist of the human orphan G-protein-coupled receptor GPR109b, with the pEC50 of 6.4. GPR109 receptor agonist-1 can be used for the research of cardio-metabolic diseases[1].

S1p receptor agonist 1

MBS131621-100mg 100mg
EUR 1495

EP4 receptor agonist 1

HY-150068 Get quote Ask for price
Description: EP4 receptor agonist 1 (compound 11) is an EP4 receptor agonist with the human pEC50 value of 6.3[1].

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